18. Protein-templated ligand discovery via the selection of DNA-encoded dynamic libraries
Yu Zhou, Wenyin Shen, Ying Gao, Jianzhao Peng, Qingrong Li, Xueying Wei, Shihao Liu, Fong Sang Lam, Joan Mayol-Llinàs, Guixian Zhao, Gang Li, Yizhou Li, Hongzhe Sun*, Yan Cao*& Xiaoyu Li*, Nature Chemistry, 2024.
17. Global profiling of functional histidines in live cells using small molecule photosensitizer and chemical probe relay labeling
Yansheng Zhai, Xinyu Zhang, Zijing Chen, Dingyuan Yan, Lin Zhu, Zhe Zhang, Xianghe Wang, Kailu Tian, Yan Huang, Xi Yang, Wen Sun, Dong Wang, Yu-Hsuan Tsai , Tuoping Luo, & Gang Li*, Nature Chemistry, 2024, Accepted. (Research Square: https://doi.org/10.21203/rs.3.rs-2981935/v1)
15. Spatiotemporal-resolved protein networks profiling with photoactivation dependent proximity labeling
Yansheng Zhai#, Xiaoyan Huang#, Keren Zhang, Yuchen Huang, Yanlong Jiang, Jingwei Cui, Zhe Zhang, Cookson Chiu, Weiye Zhong, Gang Li* . Nature Communications, 2022, 13, 4906. 【Editors' Highlights】
14. Converting Double-Stranded DNA-Encoded Libraries (DELs) to Single-Stranded Libraries for More Versatile Selections
Yuhan Gui, Clara Shania Wong, Guixian Zhao, Chao Xie, Rui Hou, Yizhou Li*, Gang Li*, and Xiaoyu Li*, ACS Omega, 2022, 7, 13, 11491–11500
13. In vivo imaging of the tumor-associated enzyme NCEH1 with a covalent PET probe
Raymond E. Moellering* Jae Won Chang, Mohammed Bhuiyan, Hsiu-Ming Tsai, Hannah J. Zhang, Gang Li, Shaghayegh Fathi, David C. McCutcheon, Lara Leoni, Richard Freifelder, Chin-Tu Chen, Angew. Chem. Int. Ed., 2020, 59(35), 15161-15165.
12. Ultrasensitive, multiplexed chemoproteomic profiling with soluble activity-dependent proximity ligation
Gang Li, Mark A. Eckert, Jae W. Chang, Jeffrey E. Montgomery, Agnieszka Chryplewicz, Ernest Lengyel, Raymond E. Moellering*, Proc. Natl. Acad. Sci. U.S.A. 2019, 116, 21493-21500.
11. A concise, modular antibody-oligonucleotide conjugation strategy based on disuccinimidyl ester activation chemistry
Gang Li, Raymond E. Moellering*, ChemBioChem, 2019, 20, 1599-1605.
10. Chemical probes for spatially resolved measurement of active enzymes in single cells
Gang Li, Raymond E. Moellering*, Methods Enzymol. 2019, 628, 243-262.
9. Proteomics reveals NNMT as a master metabolic regulator of cancer associated fibroblasts
Mark A. Eckert, Fabian Coscia, Agnieszka Chryplewicz, Jae W. Chang, Kyle M. Hernandez, Shawn Pan, Samantha M. Tienda, Dominik A. Nahotko, Gang Li, Ivana Blaženović, Ricardo R. Lastra, Marion Curtis, S. Diane Yamada, Ruth Perets, Stephanie M. McGregor, Jorge Andrade, Oliver Fiehn, Raymond E. Moellering, Matthias Mann, Ernst Lengyel*, Nature, 2019, 569, 723-728
8. An activity-dependent proximity ligation platform for spatially resolved quantification of active enzymes in single cells
Gang Li, Jeffrey E. Montgomery, Mark A. Eckert, Jae W. Chang, Sam M. Tienda, Ernest Lengyel, Raymond E. Moellering*, Nat. Commun.2017, 8, 1775-1787.
7. Stapled peptide inhibitors of RAB25 target context-specific phenotypes in cancer
Shreya Mitra, Jeffrey E. Montgomery, Matthew J. Kolar, Gang Li, Kang J. Jeong, Bo Peng, Gregory L. Verdine, Gordon B. Mills, Raymond E. Moellering*, Nat. Commun.2017, 8, 660-670.
Yun Zhang, Yibin Xue, Gang Li, Haosen Yuan, Tuoping Luo*, Chem. Sci. 2016, 7, 5530-5536.
5. Design, preparation, and selection of DNA-encoded dynamic libraries
Gang Li#, Wenlu Zheng#, Zitian Chen#, Yu Zhou, Yu Liu, Junrui Yang, Yanyi Huang, Xiaoyu Li*, Chem. Sci. 2015, 6, 7097-7104.
4. Novel encoding methods for DNA-templated chemical libraries
Gang Li, Wenlu Zheng, Ying Liu, Xiaoyu Li*, Curr. Opin. Chem. Biol. 2015, 26, 25-33.
3. Affinity purification in target identification: the specificity challenge
Wenlu Zheng, Gang Li, Xiaoyu Li*, Arch. Pharm. Res. 2015, 38, 1661-1685.
2. Multivalent photoaffinity probe for labeling small molecule binding proteins
Gang Li, Yu Liu, Xuerong Yu, Xiaoyu Li*, Bioconjugate Chem. 2014, 25, 1172-1180.
1. Photoaffinity labeling of small-molecule-binding proteins by DNA-templated chemistry
Gang Li, Ying Liu, Yu Liu, Li Chen, Siyu Wu, Yang Liu, Xiaoyu Li*, Angew. Chem. Int. Ed. 2013, 52, 9544-9549.
Address:Gaoke International Innovation Center, Guangming District,
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